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Cat. No. Product Name Target Signaling Pathways
TQ0318L ARRY 520 hydrochloride

KSP Cell Cycle/Checkpoint
ARRY 520 hydrochloride 是一种驱动蛋白纺锤体蛋白 (KSP) 抑制剂。它通过凋亡诱导细胞死亡,并具有有效的抗增殖活性。
T25418 Filanesib TFA

Filanesib trifluoroacetic acid,ARRY-520 TFA,ARRY 520 TFA,ARRY520 TFA

Filanesib (ARRY-520) targets the kinesin spindle protein (KSP) with potential antineoplastic activity. ARRY-520 specifically inhibits KSP (kinesin-5 or Eg5), resulting in activation of the spindle assembly checkpoint, induction of cell cycle arrest during
T10373 (R)-Filanesib

(R)-ARRY-520

Others Others
(R)-Filanesib is the R-enantiomer of ARRY-520. (R)-Filanesib is a synthetic kinesin spindle protein (KSP) inhibitor (IC50: 6 nM).
TQ0318 Filanesib

ARRY-520,ARRY 520

KSP Cell Cycle/Checkpoint
Filanesib (ARRY 520) 是一种选择性的驱动蛋白纺锤体蛋白(KSP)的抑制剂(IC50 = 6 nM),具有强大的抗增殖活性。

化合物

ARRY 520 hydrochloride
Cat.No: TQ0318L
Synonym:
Target: KSP
Filanesib TFA
Cat.No: T25418
Synonym: Filanesib trifluoroacetic acid,ARRY-520 TFA,ARRY 520 TFA,ARRY520 TFA
Target:
(R)-Filanesib
Cat.No: T10373
Synonym: (R)-ARRY-520
Target: Others
Filanesib
Cat.No: TQ0318
Synonym: ARRY-520,ARRY 520
Target: KSP
TargetMol Loading
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